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Kinase Drug Discovery (Rsc Drug Discovery)

by Richard A. Ward, Frederick Goldberg, David P. Rotella and David E. Thurston

KinaseInhBoook


Available in Dec 2011.

Visit our bookshelf for more books on Kinases and Kinase Inhibitors or pre-order this book today




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Articles of Interest
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# Article Title Author Hits
1 KKB Hot Article: Indirubin derivatives as potent FLT3 inhibitors with anti-proliferative activity of acute myeloid leukemic cells KKB 354
2 KKB Hot Article: Phenylaminopyrimidines as inhibitors of Janus kinases (JAKs). KKB 297
3 KKB Hot Article: 2,4-Diaminopyrimidine MK2 inhibitors. Part II: Structure-based inhibitor optimization. KKB 294
4 KKB Hot Article: Substituted 2-arylbenzothiazoles as kinase inhibitors: hit-to-lead optimization. KKB 276
5 KKB Hot Article: Targeting cancer with small molecule kinase inhibitors KKB 339
6 KKB Hot Article: Discovery of 4-morpholino-6-aryl-1H-pyrazolo[3,4-d]pyrimidines as highly potent and selective ATP-competitive inhibitors of the mammalian target of rapamycin (mTOR): optimization of the 6-aryl substituent. KKB 331
7 KKB Hot Article: Discovery of pyrimidine benzimidazoles as Src-family selective Lck inhibitors. Part II. KKB 285
8 KKB Hot Article: AC220 is a uniquely potent and selective inhibitor of FLT3 for the treatment of acute myeloid leukemia (AML). KKB 452
9 KKB Hot Article: BIBF 1120: triple angiokinase inhibitor with sustained receptor blockade and good antitumor efficacy KKB 313
10 KKB Hot Article: Selectivity and potency of cyclin-dependent kinase inhibitors KKB 289
 
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